SymbolRLAY
NameRELAY THERAPEUTICS, INC.
SectorHEALTH CARE
RegionNorth America
IndustryBiotechnology: Biological Products (No Diagnostic Substances)
Address399 BINNEY STREET,2ND FLOOR, CAMBRIDGE, Massachusetts, 02139, United States
Telephone+1 617 370-8837
Fax
Email
Websitehttps://www.relaytx.com
IncorporationUNDEFINED
Incorporated On
Employees
Fiscal Year
Public Since
ExchangesNASDAQ
Auditor
Audit StatusNOT PROVIDED
Reporting Status
CIK0001812364
Description

Relay Therapeutics Inc is a clinical-stage, precision medicines company transforming the drug discovery process with an initial focus on enhancing small molecule therapeutic discovery in targeted oncology. The company is advancing its pipeline of medicines to address targets in precision oncology, including its lead product candidates, RLY-4008 and RLY-1971, as well as its PI3Ka mutant selective program, known as the RLY-PI3K1047 program. Its initiated a Phase 1 clinical trial for RLY-1971 in patients with advanced solid tumors in the first quarter of 2020 and a first-in-human clinical trial of RLY-4008 enriched for patients with advanced solid tumors having oncogenic FGFR2 alterations in the third quarter of 2020.

Additional info from NASDAQ:
Relay Therapeutics Inc is a clinical-stage, precision medicines company transforming the drug discovery process with an initial focus on enhancing small molecule therapeutic discovery in targeted oncology. The company is advancing its pipeline of medicines to address targets in precision oncology, including its lead product candidates, RLY-4008 and RLY-1971, as well as its PI3Ka mutant selective program, known as the RLY-PI3K1047 program. Its initiated a Phase 1 clinical trial for RLY-1971 in patients with advanced solid tumors in the first quarter of 2020 and a first-in-human clinical trial of RLY-4008 enriched for patients with advanced solid tumors having oncogenic FGFR2 alterations in the third quarter of 2020.

2026-08-18 20:17

Patel Sanjiv 🔴 sold 48.2K shares of Relay Therapeutics, Inc. (RLAY) at $20.33 Transaction Date: Aug 17, 2026 | Filing ID: 355502

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2026-08-18 20:16

Catinazzo Thomas 🔴 sold 17.7K shares of Relay Therapeutics, Inc. (RLAY) at $19.74 Transaction Date: Aug 14, 2026 | Filing ID: 355493

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2026-08-14 17:17

New Form SCHEDULE 13G/A - Relay Therapeutics, Inc. <b>Filed:</b> 2026-08-14 <b>AccNo:</b> 0001831942-26-000036 <b>Size:</b> 14 KB

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2026-08-10 17:00

New Form SCHEDULE 13G/A - Relay Therapeutics, Inc. <b>Filed:</b> 2026-08-10 <b>AccNo:</b> 0001193125-26-342308 <b>Size:</b> 10 KB

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2026-08-07 12:20

New Form SCHEDULE 13G/A - Relay Therapeutics, Inc. <b>Filed:</b> 2026-08-07 <b>AccNo:</b> 0000315066-26-002255 <b>Size:</b> 11 KB

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2026-08-06 20:05

Relay Therapeutics Reports Second Quarter 2026 Financial Results and Corporate Updates

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2026-07-31 20:05

📋 SEKAR KATHIRESAN (Director) plans to sell 30K shares of RELAY THERAPEUTICS, INC. (at $18.79 each, total $564K) Filed: Jul 31, 2026 | ID: 007457

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2026-07-30 20:13

Catinazzo Thomas 🔴 sold 1.5K shares of Relay Therapeutics, Inc. (RLAY) at $18.61 Transaction Date: Jul 28, 2026 | Filing ID: 326144

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2026-07-30 20:13

Rahmer Peter 🔴 sold 748 shares of Relay Therapeutics, Inc. (RLAY) at $18.61 Transaction Date: Jul 28, 2026 | Filing ID: 326142

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2026-07-30 20:12

Bergstrom Donald A 🔴 sold 2.2K shares of Relay Therapeutics, Inc. (RLAY) at $18.61 Transaction Date: Jul 28, 2026 | Filing ID: 326137

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Trial ID Title Phase Indication Status Start Date Completion Date Source
NCT07584226 A First-in-human Study of RLY-8161 in Advanced NRAS-Mutant Solid Tumors Phase1 Advanced NRAS-Mutant Melanoma Recruiting 2026-03-09 2029-12-31 ClinicalTrials.gov
NCT06982521 Phase 3 Study of RLY-2608 + Fulvestrant vs Capivasertib + Fulvestrant as Treatm… Phase3 PIK3CA Mutation Recruiting 2025-08-26 2031-12-31 ClinicalTrials.gov
NCT06789913 A Phase 2 Study of Mutant-selective PI3Kα Inhibitor, RLY-2608, in Adults and Ch… Phase2 PIK3CA-Related Overgrowth Spectrum (PROS) Recruiting 2025-06-13 2031-10-01 ClinicalTrials.gov
NCT05759949 First-in-Human Study of RLY-5836 in Advanced Breast Cancer and Other Solid Tumo… Phase1 PIK3CA Mutation Completed 2023-03-29 2025-04-11 ClinicalTrials.gov
NCT05216432 First-in-Human Study of Mutant-selective PI3Kα Inhibitor, RLY-2608, as a Single… Phase1 PIK3CA Mutation Recruiting 2021-12-08 2027-04-30 ClinicalTrials.gov
NCT04622527 A Study to Assess Virtual Reality by Healthcare Providers: A Pilot Study Na Anxiety Completed 2021-01-01 2022-12-01 ClinicalTrials.gov
Total clinical trials: 6
Product Name Type Development Stage Therapeutic Area Study Status Trial ID
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Fulvestrant Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Capivasertib Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Zovegalisib Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Fulvestrant Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Capivasertib Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-2608 Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-8161 Other Phase PHASE1 Advanced NRAS-Mutant Melanoma RECRUITING NCT07584226
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Fulvestrant Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Capivasertib Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-2608 Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-8161 Other Phase PHASE1 Advanced NRAS-Mutant Melanoma RECRUITING NCT07584226
RLY-8161 Other Phase PHASE1 NRAS Mutation RECRUITING NCT07584226
RLY-8161 Other Phase PHASE1 NRAS Mutation RECRUITING NCT07584226
RLY-8161 Other Phase PHASE1 NRAS Mutation RECRUITING NCT07584226
RLY-8161 Other Phase PHASE1 NRAS Mutation RECRUITING NCT07584226
RLY-8161 Other Phase PHASE1 NRAS Mutation RECRUITING NCT07584226
RLY-8161 Other Phase PHASE1 NRAS Mutation RECRUITING NCT07584226
Fulvestrant Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Capivasertib Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-2608 Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Fulvestrant Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Capivasertib Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-2608 Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Fulvestrant Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Capivasertib Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-2608 Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Fulvestrant Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Capivasertib Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-2608 Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Fulvestrant Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Capivasertib Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-2608 Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Random assigned paradigm viewing order Other Approved Anxiety COMPLETED NCT04622527
Abemaciclib Other Phase PHASE1 PIK3CA Mutation COMPLETED NCT05759949
Ribociclib Other Phase PHASE1 PIK3CA Mutation COMPLETED NCT05759949
Palbociclib Other Phase PHASE1 PIK3CA Mutation COMPLETED NCT05759949
Fulvestrant Other Phase PHASE1 PIK3CA Mutation COMPLETED NCT05759949
RLY-5836 Other Phase PHASE1 PIK3CA Mutation COMPLETED NCT05759949
PF-07220060 300 mg Other Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
PF-07220060 100mg Other Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
Ribociclib 600mg Other Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
Ribociclib 400mg Other Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
Palbociclib 125mg Other Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
Fulvestrant Other Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
RLY-2608 Other Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
Fulvestrant Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Capivasertib Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-2608 Other Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Placebo Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
RLY-2608 Other Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Capivasertib DRUG Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Placebo DRUG Phase PHASE2 PIK3CA-Related Overgrowth Spectrum (PROS) RECRUITING NCT06789913
Abemaciclib DRUG Phase PHASE1 PIK3CA Mutation COMPLETED NCT05759949
Ribociclib DRUG Phase PHASE1 PIK3CA Mutation COMPLETED NCT05759949
Palbociclib DRUG Phase PHASE1 PIK3CA Mutation COMPLETED NCT05759949
RLY-5836 DRUG Phase PHASE1 PIK3CA Mutation COMPLETED NCT05759949
PF-07220060 300 mg DRUG Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
PF-07220060 100mg DRUG Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
Ribociclib 600mg DRUG Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
Ribociclib 400mg DRUG Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
Palbociclib 125mg DRUG Phase PHASE1 PIK3CA Mutation RECRUITING NCT05216432
Fulvestrant DRUG Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
RLY-2608 DRUG Phase PHASE3 PIK3CA Mutation RECRUITING NCT06982521
Random assigned paradigm viewing order OTHER Approved Anxiety COMPLETED NCT04622527
Total products: 100